Synthesis and antimicrobial activity of tryptanthrin adducts with ketones
- 作者: Deryabin P.I.1, Moskovkina T.V.1, Shevchenko L.S.2, Kalinovskii A.I.2
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隶属关系:
- Far Eastern Federal University
- Elyakov Pacific Institute of Bioorganic Chemistry, Far Eastern Branch
- 期: 卷 53, 编号 3 (2017)
- 页面: 418-422
- 栏目: Article
- URL: https://journal-vniispk.ru/1070-4280/article/view/215946
- DOI: https://doi.org/10.1134/S1070428017030174
- ID: 215946
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详细
Reactions of tryptanthrin with acetone, cyclopentanone, hexan-2-one, 4-methylpentan-2-one, 4-hydroxy-4-methylpentan-2-one, cyclohexanone, and butan-2-one in the presence of potassium carbonate afforded racemic phaitanthrin A and other addition products to the ketone group of tryptanthrin with high yields. Thermal dissociation, some chemical transformations, and antimicrobial activity of some adducts were studied, and inhibitory effect against gram-positive bacteria was found for particular derivatives.
作者简介
P. Deryabin
Far Eastern Federal University
Email: moskovkinataisiya@mail.ru
俄罗斯联邦, ul. Sukhanova 8, Vladivostok, 690091
T. Moskovkina
Far Eastern Federal University
编辑信件的主要联系方式.
Email: moskovkinataisiya@mail.ru
俄罗斯联邦, ul. Sukhanova 8, Vladivostok, 690091
L. Shevchenko
Elyakov Pacific Institute of Bioorganic Chemistry, Far Eastern Branch
Email: moskovkinataisiya@mail.ru
俄罗斯联邦, pr. 100 let Vladivostoku 159, Vladivostok, 690022
A. Kalinovskii
Elyakov Pacific Institute of Bioorganic Chemistry, Far Eastern Branch
Email: moskovkinataisiya@mail.ru
俄罗斯联邦, pr. 100 let Vladivostoku 159, Vladivostok, 690022
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