Отправить статью по E-mail Solvent-Free Synthesis, ADME Prediction, and Evaluation of Antibacterial Activity of Novel Sulfonamide Derivatives
- Авторы: Rafiee Pour Z.1, Nazifi S.M.2, Afshari Safavi A.3, Nazifi Z.S.1, Massah A.R.1,4
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Учреждения:
- Department of Chemistry, Shahreza Branch
- Department of Medicinal Chemistry, School of Pharmacy and Pharmaceutical Sciences
- Student Research Committee, School of Health
- Razi Chemistry Research Center, Shahreza Branch
- Выпуск: Том 55, № 6 (2019)
- Страницы: 852-859
- Раздел: Review
- URL: https://journal-vniispk.ru/1070-4280/article/view/220770
- DOI: https://doi.org/10.1134/S1070428019060162
- ID: 220770
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Аннотация
A series of novel sulfonamides containing a 2-amino-1,3-thiazole fragment have been synthesized using a simple and efficient method under solvent-free conditions. The obtained N-(4-sulfamoyl-1,3-thiazol-2-yl)-4-nitrobenzamides were evaluated for their antibacterial activity against S. aureus and E. coli, and in silico ADME prediction was performed to find biological behavior.
Об авторах
Z. Rafiee Pour
Department of Chemistry, Shahreza Branch
Email: massah@iaush.ac.ir
Иран, Shahreza, Isfahan
S. Nazifi
Department of Medicinal Chemistry, School of Pharmacy and Pharmaceutical Sciences
Email: massah@iaush.ac.ir
Иран, Isfahan
A. Afshari Safavi
Student Research Committee, School of Health
Email: massah@iaush.ac.ir
Иран, Isfahan
Z. Nazifi
Department of Chemistry, Shahreza Branch
Email: massah@iaush.ac.ir
Иран, Shahreza, Isfahan
A. Massah
Department of Chemistry, Shahreza Branch; Razi Chemistry Research Center, Shahreza Branch
Автор, ответственный за переписку.
Email: massah@iaush.ac.ir
Иран, Shahreza, Isfahan; Shahreza, Isfahan
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