Antiproliferative activity of ruthenium and osmium clusters with phosphine ligands


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Аннотация

New ruthenium and osmium carbonyl clusters with 1,3,5-triaza-7-phosphatricyclo-[3.3.1.13.7]decane and 3,7-diacetyl-1,3,7-triaza-5-phosphabicyclo[3.3.1]nonane ligands were synthesized using Me3NO as an initiator. The data on antiproliferative activity of new compounds against ovarian carcinoma cell cultures A2780 (cisplatin-sensitive) and A2780cisR (cisplatin-resistant) are reported. The dependence of cytotoxicity on the number of phosphine ligands was demonstrated.

Авторлар туралы

A. Nazarov

Department of Chemistry, M. V. Lomonosov Moscow State University

Хат алмасуға жауапты Автор.
Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991

Yu. Nosova

Department of Chemistry, M. V. Lomonosov Moscow State University

Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991

O. Mikhalev

Department of Chemistry, M. V. Lomonosov Moscow State University

Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991

O. Kovaleva

I. M. Sechenov First Moscow State Medical University

Email: nazarov@med.chem.msu.ru
Ресей, Build. 2, 8 ul. Trubetskaya, Moscow, 119991

P. Dyson

Swiss Federal Institute of Technology in Lausanne

Email: nazarov@med.chem.msu.ru
Швейцария, Lausanne

E. Milaeva

Department of Chemistry, M. V. Lomonosov Moscow State University

Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991

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