Antiproliferative activity of ruthenium and osmium clusters with phosphine ligands
- Авторлар: Nazarov A.A.1, Nosova Y.N.1, Mikhalev O.V.1, Kovaleva O.N.2, Dyson P.J.3, Milaeva E.R.1
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Мекемелер:
- Department of Chemistry, M. V. Lomonosov Moscow State University
- I. M. Sechenov First Moscow State Medical University
- Swiss Federal Institute of Technology in Lausanne
- Шығарылым: Том 65, № 2 (2016)
- Беттер: 546-549
- Бөлім: Full Articles
- URL: https://journal-vniispk.ru/1066-5285/article/view/237279
- DOI: https://doi.org/10.1007/s11172-016-1335-x
- ID: 237279
Дәйексөз келтіру
Аннотация
New ruthenium and osmium carbonyl clusters with 1,3,5-triaza-7-phosphatricyclo-[3.3.1.13.7]decane and 3,7-diacetyl-1,3,7-triaza-5-phosphabicyclo[3.3.1]nonane ligands were synthesized using Me3NO as an initiator. The data on antiproliferative activity of new compounds against ovarian carcinoma cell cultures A2780 (cisplatin-sensitive) and A2780cisR (cisplatin-resistant) are reported. The dependence of cytotoxicity on the number of phosphine ligands was demonstrated.
Авторлар туралы
A. Nazarov
Department of Chemistry, M. V. Lomonosov Moscow State University
Хат алмасуға жауапты Автор.
Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991
Yu. Nosova
Department of Chemistry, M. V. Lomonosov Moscow State University
Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991
O. Mikhalev
Department of Chemistry, M. V. Lomonosov Moscow State University
Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991
O. Kovaleva
I. M. Sechenov First Moscow State Medical University
Email: nazarov@med.chem.msu.ru
Ресей, Build. 2, 8 ul. Trubetskaya, Moscow, 119991
P. Dyson
Swiss Federal Institute of Technology in Lausanne
Email: nazarov@med.chem.msu.ru
Швейцария, Lausanne
E. Milaeva
Department of Chemistry, M. V. Lomonosov Moscow State University
Email: nazarov@med.chem.msu.ru
Ресей, Build. 3, 1 Leninskie Gory, Moscow, 119991
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